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BRS-3 agonist Compound A racemate
CAS No. ——
BRS-3 agonist Compound A racemate( —— )
Catalog No. M17036 CAS No. ——
A potent, selective, orally active bombesin receptor subtype-3 (BRS-3) agonist.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
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Biological Information
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Product NameBRS-3 agonist Compound A racemate
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NoteResearch use only, not for human use.
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Brief DescriptionA potent, selective, orally active bombesin receptor subtype-3 (BRS-3) agonist.
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DescriptionA potent, selective, orally active bombesin receptor subtype-3 (BRS-3) agonist with EC50 of 270/130 nM for human/rat BRS-3, respectively; displays no activity against GRPR (BRS-1) and NMBR (BRS-2) (EC50>10 uM).
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayGPCR/G Protein
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TargetBombesin Receptor
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RecptorBombesin Receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number——
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Formula Weight428.532
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Molecular FormulaC27H28N2O3
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Purity>98% (HPLC)
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Solubility——
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SMILES——
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Chemical Name6-benzyl-N-tert-butyl-9-methoxy-7-oxo-6,7-dihydro-5H-dibenzo[c,e]azepine-5-carboxamide
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Nio Y, et al. Endocrinology. 2017 May 1;158(5):1298-1313.
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Bombesin
Bombesin is a 14-amino acid peptide originally isolated from the skin of the European fire-bellied toad (Bombina bombina). It has two known homologs in mammals called neuromedin B and gastrin-releasing peptide.
